Consorzio Interuniversitario per lo sviluppo dei Sistemi a Grande Interfase
Center for Colloid and Surface Science

PUBLICATIONS

Here you can find the updated list of all the publications of CSGI members and affilated staff. Please note that the only publications listed here are those published after the affilation of each member. If you are interested in the whole bibliography of CSGI members, including articles and books published before affilation to CSGI, please refer to academic research databases, such as Scopus, Web Of Science, Google Scholar, ect.

You can use the search bar below to filter the publication list.

2025

Redesigning oxazolidinones as carbonic anhydrase inhibitors against vancomycin-resistant enterococci

- Ammara A. - Giovannuzzi S. - Bonardi A. - Abutaleb N.S. - Abouelkhair A.A. - Flaherty D.P. - Seleem M.N. - Clemente Capasso - Gratteri P. - Nocentini Alessio - Supuran C.T.
European Journal of Medicinal Chemistry

Exploring aliphatic sulfonamides as multiclass inhibitors of the carbonic anhydrases from the pathogen bacterium Vibrio cholerae

- Paoletti N. - Giovannuzzi S. - Bonardi A. - De Luca V. - Clemente Capasso - Nocentini Alessio - Gratteri P. - Supuran C.T.
Archiv der Pharmazie

2024

Synthesis and investigation of selective human carbonic anhydrase IX, XII inhibitors using coumarins bearing a sulfonamide or biotin moiety

- Begines P. - Bonardi A. - Giovannuzzi S. - Nocentini Alessio - Gratteri P. - De Luca V. - González-Bakker A. - Padrón J.M. - Clemente Capasso - Supuran C.T.
Chemico-Biological Interactions

Hydrogen Sulfide-Releasing Carbonic Anhydrase Inhibitors Effectively Suppress Cancer Cell Growth

- Bonardi A. - Nocentini Alessio - de Luca V. - Clemente Capasso - Elkaeed E.B. - Eldehna W.M. - Supuran C.T.
International Journal of Molecular Sciences

Development of Penicillin-Based Carbonic Anhydrase Inhibitors Targeting Multidrug-Resistant Neisseria gonorrhoeae

- Bonardi A. - Nocentini Alessio - Giovannuzzi S. - Paoletti N. - Ammara A. - Bua S. - Abutaleb N.S. - Abdelsattar A.S. - Clemente Capasso - Gratteri P. - Flaherty D.P. - Seleem M.N. - Supuran C.T.
Journal of Medicinal Chemistry

Leveraging SARS-CoV-2 Main Protease (Mpro) for COVID-19 Mitigation with Selenium-Based Inhibitors

- De Luca V. - Angeli A. - Nocentini Alessio - Gratteri P. - Pratesi S. - Tanini D. - Carginale V. - Capperucci A. - Supuran C.T. - Clemente Capasso
International journal of molecular sciences

2023

CD73 Inhibitors as Antitumor Agents

- Clemente Capasso - Nocentini Alessio - Supuran C.T.
Topics in Medicinal Chemistry

Aryl derivatives of 3H-1,2-benzoxaphosphepine 2-oxides as inhibitors of cancer-related carbonic anhydrase isoforms IX and XII

- Balašova A. - Pustenko A. - Nocentini Alessio - Daniela Vullo - Supuran C.T. - Žalubovskis R.
Journal of Enzyme Inhibition and Medicinal Chemistry

2022

Biochemical, structural, and computational studies of a γ-carbonic anhydrase from the pathogenic bacterium Burkholderia pseudomallei

- Di Fiore A. - De Luca V. - Langella E. - Nocentini Alessio - Buonanno M. - Monti S.M. - Supuran C.T. - Clemente Capasso - De Simone G.
Computational and Structural Biotechnology Journal

Coumarins inhibit η-class carbonic anhydrase from Plasmodium falciparum

- Giovannuzzi S. - De Luca V. - Nocentini Alessio - Clemente Capasso - Supuran C.T.
Journal of Enzyme Inhibition and Medicinal Chemistry

Inhibition studies of bacterial α-carbonic anhydrases with phenols

- Giovannuzzi S. - Hewitt C.S. - Nocentini Alessio - Clemente Capasso - Costantino G. - Flaherty D.P. - Supuran C.T.
Journal of Enzyme Inhibition and Medicinal Chemistry

Coumarins effectively inhibit bacterial α-carbonic anhydrases

- Giovannuzzi S. - Hewitt C.S. - Nocentini Alessio - Clemente Capasso - Flaherty D.P. - Supuran C.T.
Journal of Enzyme Inhibition and Medicinal Chemistry

2021

Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase

- Nocentini Alessio - Angeli A. - Carta F. - Winum J.Y. - Zalubovskis R. - Carradori S. - Clemente Capasso - Donald W.A. - Supuran C.T.
Journal of Enzyme Inhibition and Medicinal Chemistry

Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors

- Angeli A. - Carta F. - Nocentini Alessio - Winum J.Y. - Zalubovskis R. - Onnis V. - Eldehna W.M. - Clemente Capasso - Carradori S. - Donald W.A. - Dedhar S. - Supuran C.T.
Biophysical Journal

An overview on the recently discovered iota-carbonic anhydrases

- Nocentini Alessio - Supuran C.T. - Clemente Capasso
Journal of Enzyme Inhibition and Medicinal Chemistry

Development of novel quinoline-based sulfonamides as selective cancer-associated carbonic anhydrase isoform ix inhibitors

- Shaldam M. - Nocentini Alessio - Elsayed Z.M. - Ibrahim T.M. - Salem R. - El-Domany R.A. - Clemente Capasso - Supuran C.T. - Eldehna W.M.
International Journal of Molecular Sciences

Selective inhibition of helicobacter pylori carbonic anhydrases by carvacrol and thymol could impair biofilm production and the release of outer membrane vesicles

- Grande R. - Carradori S. - Puca V. - Vitale I. - Angeli A. - Nocentini Alessio - Bonardi A. - Gratteri P. - Lanuti P. - Bologna G. - Simeone P. - Clemente Capasso - De Luca V. - Supuran C.T.
International Journal of Molecular Sciences

Anion inhibition studies of the Zn(II)-bound ι-carbonic anhydrase from the Gram-negative bacterium Burkholderia territorii

- Petreni A. - De Luca V. - Scaloni A. - Nocentini Alessio - Clemente Capasso - Supuran C.T.
Journal of Enzyme Inhibition and Medicinal Chemistry

Development of novel benzofuran-based SLC-0111 analogs as selective cancer-associated carbonic anhydrase isoform IX inhibitors

- Shaldam M. - Eldehna W.M. - Nocentini Alessio - Elsayed Z.M. - Ibrahim T.M. - Salem R. - El-Domany R.A. - Clemente Capasso - Abdel-Aziz H.A. - Supuran C.T.
European Journal of Medicinal Chemistry

2020

Carbonic anhydrase inhibitors targeting metabolism and tumor microenvironment

- Angeli A. - Carta F. - Nocentini Alessio - Winum J.Y. - Zalubovskis R. - Akdemir A. - Onnis V. - Eldehna W.M. - Clemente Capasso - Simone G.D. - Monti S.M. - Carradori S. - Donald W.A. - Dedhar S. - Supuran C.T.
Metabolites

Phosphonamidates are the first phosphorus-based zinc binding motif to show inhibition of β-class carbonic anhydrases from bacteria, fungi, and protozoa

- Alissa S.A. - Alghulikah H.A. - Alothman Z.A. - Osman S.M. - Del Prete S. - Clemente Capasso - Nocentini Alessio - Supuran C.T.
Journal of Enzyme Inhibition and Medicinal Chemistry

Inhibition survey with phenolic compounds against the δ- and η-class carbonic anhydrases from the marine diatom thalassiosira weissflogii and protozoan Plasmodium falciparum

- Alissa S.A. - Alghulikah H.A. - ALOthman Z.A. - Osman S.M. - Del Prete S. - Clemente Capasso - Nocentini Alessio - Supuran C.T.
Journal of Enzyme Inhibition and Medicinal Chemistry

Activation studies of the β-carbonic anhydrases from Escherichia coli with amino acids and amines

- Nocentini Alessio - Del Prete S. - Mastrolorenzo M.D. - Donald W.A. - Clemente Capasso - Supuran C.T.
Journal of Enzyme Inhibition and Medicinal Chemistry

"a Sweet Combination": Developing Saccharin and Acesulfame K Structures for Selectively Targeting the Tumor-Associated Carbonic Anhydrases IX and XII

- Bua S. - Lomelino C. - Murray A.B. - Osman S.M. - Alothman Z.A. - Murat Bozdag - Abdel-Aziz H.A. - Eldehna W.M. - McKenna R. - Nocentini Alessio - Supuran C.T.
Journal of Medicinal Chemistry

Discovery of New 1,1′-Biphenyl-4-sulfonamides as Selective Subnanomolar Human Carbonic Anhydrase II Inhibitors

- La Regina G. - Puxeddu M. - Nalli M. - Daniela Vullo - Gratteri P. - Supuran C.T. - Nocentini Alessio - Silvestri R.
ACS Medicinal Chemistry Letters

Anion inhibition studies of the beta-carbonic anhydrase from Escherichia coli

- Del Prete S. - De Luca V. - Nocentini Alessio - Scaloni A. - Mastrolorenzo M.D. - Supuran C.T. - Clemente Capasso
Molecules

Structural and biochemical characterization of novel carbonic anhydrases from Phaeodactylum tricornutum Jin Shengyang

- Jin S. - Daniela Vullo - Bua S. - Nocentini Alessio - Supuran C.T. - Gao Y.G.
Acta Crystallographica Section D: Structural Biology

Halogenated isophthalamides and dipicolineamides: The role of the halogen substituents in the anion binding properties

- Picci G. - Bazzicalupi C. - Coles S.J. - Gratteri P. - Isaia F. - Vito Lippolis - Montis R. - Sergio Murgia - Nocentini Alessio - Orton J.B. - Claudia Caltagirone
Dalton Transactions

Benzoxaboroles: New Potent Inhibitors of the Carbonic Anhydrases of the Pathogenic Bacterium Vibrio cholerae

- Bonardi A. - Nocentini Alessio - Cadoni R. - Del Prete S. - Dumy P. - Clemente Capasso - Gratteri P. - Supuran C.T. - Winum J.Y.
ACS Medicinal Chemistry Letters

2019

Synthesis and evaluation of carbonic anhydrase inhibitors with carbon monoxide releasing properties for the management of rheumatoid arthritis

- Berrino E. - Milazzo L. - Micheli L. - Daniela Vullo - Angeli A. - Murat Bozdag - Nocentini Alessio - Menicatti M. - Bartolucci G. - Di Cesare Mannelli L. - Ghelardini C. - Supuran C.T. - Carta F.
Journal of Medicinal Chemistry

Phaeodactylum tricornutum as a model organism for testing the membrane penetrability of sulphonamide carbonic anhydrase inhibitors

- Rogato A. - Del Prete S. - Nocentini Alessio - Carginale V. - Supuran C. - Clemente Capasso
Journal of Enzyme Inhibition and Medicinal Chemistry

Extending the γ-class carbonic anhydrases inhibition profiles with phenolic compounds

- Nocentini Alessio - Osman S.M. - Del Prete S. - Clemente Capasso - ALOthman Z.A. - Supuran C.T.
Bioorganic Chemistry

2018

2017

Dithiocarbamates effectively inhibit the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa

- Daniela Vullo - Del Prete S. - Nocentini Alessio - Osman S.M. - AlOthman Z. - Clemente Capasso - Murat Bozdag - Carta F. - Gratteri P. - Supuran C.T.
Bioorganic and Medicinal Chemistry

Inhibition of Malassezia globosa carbonic anhydrase with phenols

- Entezari Heravi Y. - Bua S. - Nocentini Alessio - Del Prete S. - Saboury A.A. - Sereshti H. - Clemente Capasso - Gratteri P. - Supuran C.T.
Bioorganic and Medicinal Chemistry

Inhibition of the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa with monothiocarbamates

- Nocentini Alessio - Daniela Vullo - Del Prete S. - Osman S. - Alasmary F. - AlOthman Z. - Clemente Capasso - Carta F. - Gratteri P. - Supuran C.
Journal of Enzyme Inhibition and Medicinal Chemistry

Lipoyl-Homotaurine Derivative (ADM-12) Reverts Oxaliplatin-Induced Neuropathy and Reduces Cancer Cells Malignancy by Inhibiting Carbonic Anhydrase IX (CAIX)

- Fragai M. - Comito G. - Di Cesare Mannelli L. - Gualdani R. - Calderone V. - Louka A. - Barbara Richichi - Francesconi O. - Angeli A. - Nocentini Alessio - Gratteri P. - Chiarugi P. - Ghelardini C. - Francesco Tadini Buoninsegni - Supuran C.T. - Nativi C.
Journal of Medicinal Chemistry

Benzoxaboroles as Efficient Inhibitors of the β-Carbonic Anhydrases from Pathogenic Fungi: Activity and Modeling Study

- Nocentini Alessio - Cadoni R. - Del Prete S. - Clemente Capasso - Dumy P. - Gratteri P. - Supuran C.T. - Winum J.Y.
ACS Medicinal Chemistry Letters

2016

N-Nitrosulfonamides: A new chemotype for carbonic anhydrase inhibition

- Nocentini Alessio - Daniela Vullo - Bartolucci G. - Supuran C.T.
Bioorganic and Medicinal Chemistry